Bisindolylmaleimide I ≥98% (by TLC)

Supplier: ENZO LIFE SCIENCES AG

Synonyms: 3-(1-(3-(Dimethylamino)propyl)-1H-indol-3-yl)-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione, 3-[1-[3-(Dimethylamino)propyl]-1H-indol-3-yl]-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione, GF 109203X

BMLEI2460001 BMLEI2460005
ENZOBMLEI2460001EA 107 GBP
ENZOBMLEI2460001 ENZOBMLEI2460005
Bisindolylmaleimide I ≥98% (by TLC)
Bisindolylmaleimide I

Potent and selective protein kinase C inhibitor which has been used effectively in platelets, Swiss 3T3 fibroblasts and macrophages. Inhibitory profile: PKC, IC50=0.02µM (inhibits α, ßI, ßII and γ subtypes with similar potency); PKA, IC50=2.0µM; phosphorylase kinase, IC50=0.7µM; insulin, EGF and PDGF receptor tyrosine kinases are not inhibited at concentrations up to 50µM.


  • PKC inhibitor


Red solid.


Soluble in dimethyl formamide or DMSO (10mg/ml, warm to 40°C and vortex well). 

Formula: C₂₅H₂₄N₄O₂
MW: 412,48 g/mol
Storage Temperature: Freezer
MDL Number: MFCD00236428
CAS Number: 133052-90-1
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